In Silico strategies for drug discovery: optimizing natural compounds from foods for therapeutic applications

Αποθηκεύτηκε σε:
Λεπτομέρειες βιβλιογραφικής εγγραφής
Εκδόθηκε σε:Discover Chemistry vol. 2, no. 1 (Dec 2025), p. 133
Κύριος συγγραφέας: Aarón, Romo-Hernández
Άλλοι συγγραφείς: Sheila, Cortazar-Moya, Julio Emmanuel, González-Pérez, Oscar, Jiménez-González, Aurelio, López-Malo, Jocksan Ismael, Morales-Camacho
Έκδοση:
Springer Nature B.V.
Θέματα:
Διαθέσιμο Online:Citation/Abstract
Full Text
Full Text - PDF
Ετικέτες: Προσθήκη ετικέτας
Δεν υπάρχουν, Καταχωρήστε ετικέτα πρώτοι!

MARC

LEADER 00000nab a2200000uu 4500
001 3256873091
003 UK-CbPIL
022 |a 3005-1193 
024 7 |a 10.1007/s44371-025-00201-3  |2 doi 
035 |a 3256873091 
045 2 |b d20251201  |b d20251231 
100 1 |a Aarón, Romo-Hernández  |u Universidad de las Américas Puebla, Departamento de Ingeniería Química, Alimentos y Ambiental, Puebla, México (GRID:grid.440458.9) (ISNI:0000 0001 0150 5973) 
245 1 |a In Silico strategies for drug discovery: optimizing natural compounds from foods for therapeutic applications 
260 |b Springer Nature B.V.  |c Dec 2025 
513 |a Journal Article 
520 3 |a The physicochemical properties of natural chemical compounds serve as a foundation for the development of novel drugs and innovative therapies. While several databases describe properties of natural products, their applicability and data accessibility are limited. Thus, the lack of accessible data represents a significant challenge in developing drugs based on natural compounds. Although chemical properties of natural compounds can be determined experimentally, this approach requires costly materials and procedures. In silico alternatives for drug analysis and pharmaceutical design cycles represent an interesting, simpler, and less expensive option for natural compound-based drug discovery. This article examines in silico methods for the characterization, design, and optimization of natural compound-based drugs derived from food. The review focuses on how in silico-based tools, such as machine learning, computer-based mathematical modeling, homology prediction, docking, molecular dynamics, and simulated molecular evolution events, are used to optimize natural compound testing and design. The in silico bioactivity predicted properties for peptides and secondary metabolites are discussed. In silico analysis is also explored as a tool to predict the antioxidant, antidiabetic, antimicrobial, and cardiovascular effects of natural compounds from foods. The approaches here presented can help speed up the discovery and development of natural compound-based drugs for therapeutic use. 
653 |a Accessibility 
653 |a Chemical compounds 
653 |a Pharmacology 
653 |a Drug development 
653 |a Metabolites 
653 |a Drugs 
653 |a Peptides 
653 |a Machine learning 
653 |a Research & development--R&D 
653 |a Breast cancer 
653 |a Proteins 
653 |a Physicochemical properties 
653 |a Simulation 
653 |a Computers 
653 |a Food 
653 |a Molecular docking 
653 |a Homology 
653 |a Chemical properties 
653 |a Design 
653 |a Antihypertensives 
653 |a Molecular dynamics 
653 |a Design optimization 
653 |a Natural products 
700 1 |a Sheila, Cortazar-Moya  |u Universidad de las Américas Puebla, Departamento de Ingeniería Química, Alimentos y Ambiental, Puebla, México (GRID:grid.440458.9) (ISNI:0000 0001 0150 5973) 
700 1 |a Julio Emmanuel, González-Pérez  |u Universidad de las Américas Puebla, Departamento de Ingeniería Química, Alimentos y Ambiental, Puebla, México (GRID:grid.440458.9) (ISNI:0000 0001 0150 5973); Tecnológico de Monterrey, School of Engineering and Sciences, Monterrey, México (GRID:grid.419886.a) (ISNI:0000 0001 2203 4701) 
700 1 |a Oscar, Jiménez-González  |u Universidad de las Américas Puebla, Departamento de Ingeniería Química, Alimentos y Ambiental, Puebla, México (GRID:grid.440458.9) (ISNI:0000 0001 0150 5973); Universidad Popular Autónoma del Estado de Puebla, Faculty of Gastronomy, Puebla, Mexico (GRID:grid.441428.f) (ISNI:0000 0001 2184 565X) 
700 1 |a Aurelio, López-Malo  |u Universidad de las Américas Puebla, Departamento de Ingeniería Química, Alimentos y Ambiental, Puebla, México (GRID:grid.440458.9) (ISNI:0000 0001 0150 5973) 
700 1 |a Jocksan Ismael, Morales-Camacho  |u Universidad de las Américas Puebla, Departamento de Ingeniería Química, Alimentos y Ambiental, Puebla, México (GRID:grid.440458.9) (ISNI:0000 0001 0150 5973) 
773 0 |t Discover Chemistry  |g vol. 2, no. 1 (Dec 2025), p. 133 
786 0 |d ProQuest  |t Materials Science Database 
856 4 1 |3 Citation/Abstract  |u https://www.proquest.com/docview/3256873091/abstract/embedded/L8HZQI7Z43R0LA5T?source=fedsrch 
856 4 0 |3 Full Text  |u https://www.proquest.com/docview/3256873091/fulltext/embedded/L8HZQI7Z43R0LA5T?source=fedsrch 
856 4 0 |3 Full Text - PDF  |u https://www.proquest.com/docview/3256873091/fulltextPDF/embedded/L8HZQI7Z43R0LA5T?source=fedsrch